211280 Sigma-AldrichCapsazepine - CAS 138977-28-3 - Calbiochem
A competitive antagonist of Capsaicin and resiniferatoxin. Capsazepine (1 µM) blocks capsaicin (60 nM) stimulated firing of C-fibers.
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Synonyms: N-[2-(4-Chlorophenyl)ethyl]-1,3,4,5-tetrahydro-7,8-dihydroxy-2H-2-benzazepine-2-carbothioamide
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Overview
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Key Specifications Table
| CAS # | Empirical Formula |
|---|---|
| 138977-28-3 | C₁₉H₂₁N₂O₂SCl |
Products
| Catalog Number | Packaging | Qty/Pack | |
|---|---|---|---|
| 211280-10MG | Plastic ampoule | 10 mg |
| Description | |
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| Overview | A competitive antagonist of Capsaicin (Cat. No. 211274) and resiniferatoxin. Capsazepine (1 µM) blocks capsaicin (60 nM) stimulated firing of C-fibers. |
| Catalogue Number | 211280 |
| Brand Family | Calbiochem® |
| Synonyms | N-[2-(4-Chlorophenyl)ethyl]-1,3,4,5-tetrahydro-7,8-dihydroxy-2H-2-benzazepine-2-carbothioamide |
| Product Information | |
|---|---|
| CAS number | 138977-28-3 |
| ATP Competitive | N |
| Form | Off-white solid |
| Hill Formula | C₁₉H₂₁N₂O₂SCl |
| Chemical formula | C₁₉H₂₁N₂O₂SCl |
| Reversible | N |
| Structure formula Image | |
| Quality Level | MQ100 |
| Applications |
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| Biological Information | |
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| Primary Target | A competitive antagonist of Capsaicin and resiniferatoxin |
| Purity | ≥97% by HPLC |
| Physicochemical Information | |
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| Cell permeable | N |
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| Safety Information |
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| Specifications |
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| Global Trade Item Number | |
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| Catalog Number | GTIN |
| 211280-10MG | 04055977219180 |
Documentation
Capsazepine - CAS 138977-28-3 - Calbiochem SDS
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Capsazepine - CAS 138977-28-3 - Calbiochem Certificates of Analysis
| Title | Lot Number |
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| 211280 |
References
| Reference overview |
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| Fox, A.J., et al. 1995. Neuroscience 67, 741. Ellis, J.L., and Undem, B.J. 1994. J. Pharmacol. Exp. Ther. 268, 85. Walpole, C.S.J., et al. 1994. J. Med. Chem. 37, 1942. Szallasi, A., et al. 1993. J. Pharmacol. Exp. Therap. 267, 728. |