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231085 Cilostamide - CAS 68550-75-4 - Calbiochem

A cell-permeable selective inhibitor of cGMP-inhibited phosphodiesterase (PDE III; IC₅₀ = 70 nM).

Cilostamide - CAS 68550-75-4 - Calbiochem MSDS (material safety data sheet) or SDS, CoA and CoQ, dossiers, brochures and other available documents.

Synonyms: N-Cyclohexyl-N-methyl-4-(1,2-dihydro-2-oxo-6-quinolyloxy)butyramide, OPC 3689

Primary Target: PDE 3
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231085
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Overview

Replacement Information

Key Specifications Table

CAS #Empirical Formula
68550-75-4C₂₀H₂₆N₂O₃

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231085-10MG
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      Description
      OverviewA cell-permeable selective inhibitor of cGMP-inhibited phosphodiesterase (PDE III; IC50 = 70 nM).
      Catalogue Number231085
      Brand Family Calbiochem®
      SynonymsN-Cyclohexyl-N-methyl-4-(1,2-dihydro-2-oxo-6-quinolyloxy)butyramide, OPC 3689
      References
      ReferencesVerghese, M.W., et al. 1995. J. Pharmacol. Exp. Ther. 272, 1313.
      Christensen, S.B., and Trophy, T.J. 1994. Ann. Rep. Med. Chem. 29, 185.
      Tang, K.M., et al. 1994. Eur. J. Pharmacol. 268, 105.
      Product Information
      CAS number68550-75-4
      ATP CompetitiveN
      FormWhite solid
      Hill FormulaC₂₀H₂₆N₂O₃
      Chemical formulaC₂₀H₂₆N₂O₃
      ReversibleN
      Structure formula ImageStructure formula Image
      Quality LevelMQ100
      Applications
      Biological Information
      Primary TargetPDE 3
      Primary Target IC<sub>50</sub>70 nM against PDE III
      Purity≥98% by TLC
      Physicochemical Information
      Cell permeableY
      Dimensions
      Materials Information
      Toxicological Information
      Safety Information according to GHS
      Safety Information
      Product Usage Statements
      Storage and Shipping Information
      Ship Code Ambient Temperature Only
      Toxicity Standard Handling
      Storage +2°C to +8°C
      Do not freeze Ok to freeze
      Special InstructionsFollowing reconstitution, refrigerate (4°C). Stock solutions are stable for up to 6 months at 4°C.
      Packaging Information
      Transport Information
      Supplemental Information
      Specifications
      Global Trade Item Number
      Catalog Number GTIN
      231085-10MG 04055977217599

      Documentation

      Cilostamide - CAS 68550-75-4 - Calbiochem SDS

      Title

      Safety Data Sheet (SDS) 

      Cilostamide - CAS 68550-75-4 - Calbiochem Certificates of Analysis

      TitleLot Number
      231085

      References

      Reference overview
      Verghese, M.W., et al. 1995. J. Pharmacol. Exp. Ther. 272, 1313.
      Christensen, S.B., and Trophy, T.J. 1994. Ann. Rep. Med. Chem. 29, 185.
      Tang, K.M., et al. 1994. Eur. J. Pharmacol. 268, 105.
      Data Sheet

      Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

      Revision05-June-2008 RFH
      SynonymsN-Cyclohexyl-N-methyl-4-(1,2-dihydro-2-oxo-6-quinolyloxy)butyramide, OPC 3689
      DescriptionA cell-permeable selective inhibitor of cGMP-inhibited phosphodiesterase (PDE III; IC50 = 70 nM).
      FormWhite solid
      CAS number68550-75-4
      Chemical formulaC₂₀H₂₆N₂O₃
      Structure formulaStructure formula
      Purity≥98% by TLC
      SolubilityDMSO (5 mg/ml)
      Storage +2°C to +8°C
      Do Not Freeze Ok to freeze
      Special InstructionsFollowing reconstitution, refrigerate (4°C). Stock solutions are stable for up to 6 months at 4°C.
      Toxicity Standard Handling
      ReferencesVerghese, M.W., et al. 1995. J. Pharmacol. Exp. Ther. 272, 1313.
      Christensen, S.B., and Trophy, T.J. 1994. Ann. Rep. Med. Chem. 29, 185.
      Tang, K.M., et al. 1994. Eur. J. Pharmacol. 268, 105.